RWJ 63556 ( RWJ-63556 )

产品货号. M26425 CAS No. 190967-35-2

COA

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HNMR

HPLC

MSDS

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产品名称

RWJ 63556
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

RWJ 63556 是一种口服活性 COX-2 选择性/5-脂氧合酶抑制剂，具有抗炎活性。
产品描述

RWJ 63556 is an orally active inhibitor of COX-2 selective/5-lipoxygenase, shows anti-inflammatory activities.(In Vitro):RWJ 63556 is a potent leukocyte influx inhibitor over a period of 24 hr and maintains its in vitro profile on eicosanoids.(In Vivo):RWJ 63556 (1?mg/kg, i.v.) significantly inhibits the development of SP-induced oedema.
体外实验

RWJ 63556 is a potent inhibitor of leukocyte influx over a period of 24 hr and maintains its in vitro profile on eicosanoids.
体内实验

RWJ 63556 (1?mg/kg, i.v.) significantly inhibits the development of SP-induced oedema.
同义词

RWJ-63556
通路

Immunology/Inflammation
靶点

Lipoxygenase
受体

VHL
研究领域

——
适应症

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1.Pillow TH, et al. Antibody Conjugation of a Chimeric BET Degrader Enables in vivo Activity. ChemMedChem. 2019 Oct 31.

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